SCHEMBL8044481

SCHEMBL8044481

CN[C@@H]1CCc2c(cccc2OC)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 1.00
DRD3 P35462 8/20 1.00
DRD4 P21917 6/20 1.00
MTNR1A P48039 2/20 0.68
MTNR1B P49286 2/20 0.68
CA1 P00915 3/20 0.65
CA2 P00918 3/20 0.65
ACHE P22303 3/20 0.65
CHRM2 P08172 1/20 0.58
CHRM1 P11229 1/20 0.58
CHRM3 P20309 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044480 1.00 DRD2 (1.00) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL8044484 1.00 DRD2 (1.00) DRD2DRD3DRD4MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL10849302 0.98 DRD2 (0.97) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL4518779 0.89 DRD2 (0.80) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL7543876 0.89 DRD2 (0.80) DRD2DRD3DRD4MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7543024 0.88 DRD2 (0.78) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL2959295 0.88 DRD2 (0.78) DRD2DRD3DRD4MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7544278 0.88 DRD2 (0.78) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL338363 0.87 DRD2 (0.77) DRD2DRD3DRD4MTNR1AMTNR1B
SCHEMBL8394758 0.84 DRD2 (1.00) DRD2DRD3DRD4MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817767-B1 BICYCLIC AMINE DERIVATIVES AND THEIR USE AS ANTI-PSYCHOTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 2000-05-24 EP disclosed
US-6008219-A Bicyclic amine derivatives and their use as anti-psychotic agents SMITHKLINE BEECH P.L.C. (GB) 1999-12-28 US disclosed
EP-0817767-A1 BICYCLIC AMINE DERIVATIVES AND THEIR USE AS ANTI-PSYCHOTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1998-01-14 EP disclosed
WO-1996030333-A1 BICYCLIC AMINE DERIVATIVES AND THEIR USE AS ANTI-PSYCHOTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1996-10-03 WO disclosed