SCHEMBL8044740

SCHEMBL8044740

COCCCn1c(Sc2ncc([N+](=O)[O-])s2)nnc1-c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
TSHR P16473 3/20 0.48
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
TLR9 Q9NR96 3/20 0.46
AGTR1 P30556 2/20 0.46
MAPK8 P45983 5/20 0.46
MAPK9 P45984 5/20 0.46
HTT P42858 4/20 0.42
KDM4E B2RXH2 3/20 0.42
GAA P10253 2/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 5/20 0.39
ALDH1A1 P00352 3/20 0.39
S1PR4 O95977 2/20 0.39
S1PR1 P21453 2/20 0.39
MAPK1 P28482 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MIF P14174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045332 0.87 NPC1 (0.46) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8050094 0.85 NPC1 (0.44) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8032454 0.84 TSHR (0.49) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8050072 0.83 NPC1 (0.57) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8050456 0.83 RAB9A (0.45) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8044858 0.83 TSHR (0.49) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8045746 0.83 KMT2A (0.53) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8045928 0.80 TSHR (0.52) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8048102 0.79 MAPT (0.45) MEN1KMT2ATSHRNPC1RAB9A
SCHEMBL8443322 0.79 NPC1 (0.73) MEN1KMT2ANPC1RAB9ATLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed