SCHEMBL8046654

SCHEMBL8046654

O=C(Nc1cnc(Sc2nnc(-c3cccs3)n2C2CCCCC2)s1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.42
ALDH1A1 P00352 7/20 0.41
HSD17B10 Q99714 4/20 0.41
RAB9A P51151 3/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
NPSR1 Q6W5P4 4/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CYP3A4 P08684 4/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ADCY1 Q08828 1/20 0.39
GAA P10253 4/20 0.38
NPC1 O15118 2/20 0.38
HTT P42858 2/20 0.38
PPARG P37231 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NR2E3 Q9Y5X4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043654 0.84 TSHR (0.52) TSHRALDH1A1HSD17B10KDM4EHPGD
SCHEMBL8044921 0.83 ALDH1A1 (0.44) TSHRALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL8044457 0.83 HDAC6 (0.57) TSHRALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL8032459 0.81 HSD17B10 (0.49) TSHRALDH1A1HSD17B10KDM4EHPGD
SCHEMBL8045038 0.80 TSHR (0.47) TSHRALDH1A1HSD17B10KDM4EHPGD
SCHEMBL8046929 0.80 TSHR (0.52) TSHRALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL8051531 0.80 ALDH1A1 (0.45) TSHRALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL8051528 0.79 USP2 (0.45) TSHRALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL8046996 0.79 TSHR (0.45) TSHRALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL8043244 0.79 NPSR1 (0.46) TSHRALDH1A1HSD17B10KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed