SCHEMBL8047041

SCHEMBL8047041

CC(C)(C1CCN(C(=O)c2ccc(CC(F)F)c(S(C)(=O)=O)c2)CC1)S(=O)(=O)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 8/20 0.51
CYP3A4 P08684 2/20 0.51
NR1I2 O75469 1/20 0.48
HSD11B1 P28845 1/20 0.46
MGLL Q99685 3/20 0.45
PKLR P30613 1/20 0.41
PRKAA2 P54646 1/20 0.40
RORC P51449 1/20 0.39
MAPK7 Q13164 1/20 0.39
AKR1C3 P42330 1/20 0.39
SCN9A Q15858 1/20 0.38
SLC9A1 P19634 1/20 0.38
HRH1 P35367 1/20 0.38
CCR3 P51677 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040721 0.93 CACNA1B (0.53) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3036583 0.88 CACNA1B (0.54) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3025678 0.86 CACNA1B (0.55) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL8044492 0.85 CACNA1B (0.54) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3036590 0.84 CACNA1B (0.56) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3035867 0.84 CACNA1B (0.52) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3038986 0.82 CACNA1B (0.56) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3032252 0.82 CACNA1B (0.54) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3035386 0.82 HSD11B1 (0.57) CACNA1BCYP3A4NR1I2HSD11B1MGLL
SCHEMBL3035343 0.81 CACNA1B (0.60) CACNA1BCYP3A4NR1I2HSD11B1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009045382-A1 SUBSTITUTED ARYL SULFONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2009-04-09 WO disclosed