SCHEMBL8047487

SCHEMBL8047487

N#CC(CCCCCC(=O)NOC(=O)c1ccccc1)(c1ccccc1)c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 16/20 0.42
CCR1 P32246 1/20 0.37
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC9 Q9UKV0 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
CYP3A4 P08684 2/20 0.36
KCNH2 Q12809 2/20 0.36
CYP2C9 P11712 1/20 0.36
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
PGR P06401 1/20 0.35
THRB P10828 1/20 0.35
ADRB3 P13945 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044655 0.89 CYP3A4 (0.43) HDAC6CCR1HDAC3HDAC4HDAC1
SCHEMBL8049747 0.89 CYP3A4 (0.43) HDAC6CCR1HDAC3HDAC4HDAC1
SCHEMBL8052916 0.87 HDAC6 (0.41) HDAC6CCR1CYP3A4KCNH2CYP2C9
SCHEMBL8045859 0.84 HDAC6 (0.51) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL8045199 0.84 HDAC1 (0.38) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL8045631 0.84 HDAC6 (0.39) HDAC6CCR1HDAC3HDAC4HDAC1
SCHEMBL8049521 0.83 HDAC6 (0.49) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL8052908 0.82 KMT2A (0.40) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL8035617 0.82 KMT2A (0.40) HDAC6CCR1HDAC3HDAC4HDAC1
SCHEMBL8044657 0.80 CCR1 (0.43) HDAC6CCR1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed