SCHEMBL8047602

SCHEMBL8047602

CCCc1nn(C)c2c(=O)[nH]c(N(CCN3CCN(C(=O)C(C)C)CC3)CC3CCCCC3)nc12

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 19/20 0.38
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
HDAC1 Q13547 8/20 0.36
HDAC6 Q9UBN7 8/20 0.36
HDAC2 Q92769 3/20 0.35
MTOR P42345 1/20 0.35
PDE6C P51160 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047597 0.90 PDE5A (0.38) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL8042867 0.87 KDM4E (0.33)
SCHEMBL8050917 0.86 PDE5A (0.44) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL8045595 0.86 PDE5A (0.41) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL8049072 0.83 PDE5A (0.48) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL8047604 0.79 PDE5A (0.42) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL3993298 0.79 PDE5A (0.44) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL8045086 0.77 PDE5A (0.47) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL4136868 0.77 PDE5A (0.44) PDE5APDE3BPDE3AHDAC1HDAC6
SCHEMBL4117716 0.76 SIGMAR1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071707-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed