SCHEMBL8049044

SCHEMBL8049044

C/C(=C\c1ccc(F)cc1)C(=O)Nc1ccc(Cl)cc1C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.64
KDM4E B2RXH2 2/20 0.57
HSD17B10 Q99714 1/20 0.57
TRPM8 Q7Z2W7 1/20 0.55
GRIK1 P39086 1/20 0.46
SERPINE1 P05121 4/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
AKR1C4 P17516 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
GAA P10253 1/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
KCNK2 O95069 1/20 0.42
KCNK10 P57789 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8049046 1.00 DHODH (0.64) DHODHKDM4EHSD17B10TRPM8GRIK1
SCHEMBL8059517 0.92 KDM4E (0.62) DHODHKDM4EHSD17B10TRPM8SERPINE1
SCHEMBL8059511 0.92 KDM4E (0.62) DHODHKDM4EHSD17B10TRPM8SERPINE1
SCHEMBL8048932 0.90 GRIK1 (0.58) DHODHKDM4ETRPM8GRIK1NPC1
SCHEMBL8048928 0.90 GRIK1 (0.58) DHODHKDM4ETRPM8GRIK1NPC1
SCHEMBL8060345 0.89 KDM4E (0.58) DHODHKDM4EHSD17B10TRPM8SERPINE1
SCHEMBL8048963 0.89 KDM4E (0.58) DHODHKDM4EHSD17B10TRPM8GRIK1
SCHEMBL8060346 0.89 KDM4E (0.58) DHODHKDM4EHSD17B10TRPM8SERPINE1
SCHEMBL8048968 0.89 KDM4E (0.58) DHODHKDM4EHSD17B10TRPM8GRIK1
SCHEMBL8059614 0.89 DHODH (0.71) DHODHKDM4EHSD17B10TRPM8SERPINE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127392-A A MUSCLE RELAXANT FOR TREATMENT OF DISORDERS ASSOCIATED WITH SMOOTH MUSCLE CONTRACTION VIA POTASSIUM CHANNEL AND CHLORIDE CHANNEL MODULATION; INOTROPIC AGENT AMERICAN HOME PRODUCTS CORPORATION (US) 2000-10-03 US disclosed
US-6046239-A USED IN THE TREATMENT OF DISORDERS ASSOCIATED WITH SMOOTH MUSCLE CONTRACTION, VIA POTASSIUM CHANNEL AND CHLORIDE CHANNEL MODULATION SUCH AS URINARY INCONTINENCE, ASTHMA, ANGINA, PREMATURE LABOR, CONGESTIVE HEART FAILURE AMERICAN HOME PRODUCTS CORPORATION (US) 2000-04-04 US disclosed