SCHEMBL8049889

SCHEMBL8049889

CCCN(C(C)=O)C1CCN(CCC(C)(C(=O)NC(CC)c2ccccc2)c2ccc(I)c(Cl)c2)CC1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 3/20 0.68
TACR2 P21452 2/20 0.44
TACR1 P25103 2/20 0.44
CCR5 P51681 14/20 0.39
UBE2M P61081 3/20 0.38
DCUN1D1 Q96GG9 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL297453 0.93 TACR3 (0.77) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL296656 0.93 TACR3 (0.77) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL8053227 0.88 TACR3 (0.71) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL3275834 0.87 TACR3 (0.69) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL297449 0.87 TACR3 (0.68) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL296806 0.87 TACR3 (0.68) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL296859 0.87 TACR3 (0.68) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL297239 0.87 TACR3 (0.68) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL3272860 0.81 TACR3 (0.60) TACR3TACR2TACR1CCR5UBE2M
SCHEMBL296050 0.81 TACR3 (1.00) TACR3TACR2TACR1CCR5UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033995-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-03-19 WO disclosed