SCHEMBL8053227

SCHEMBL8053227

CCC(NC(=O)C(C)(CCN1CCC(N(CCO)C(C)=O)CC1)c1ccc(Cl)c(Cl)c1)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 6/20 0.71
TACR1 P25103 5/20 0.50
TACR2 P21452 4/20 0.50
UBE2M P61081 1/20 0.42
DCUN1D1 Q96GG9 1/20 0.42
CCR5 P51681 11/20 0.42
PPARG P37231 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL296656 0.95 TACR3 (0.77) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL297453 0.95 TACR3 (0.77) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL296806 0.93 TACR3 (0.68) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL297449 0.93 TACR3 (0.68) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL296859 0.92 TACR3 (0.68) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL297239 0.92 TACR3 (0.68) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL8049889 0.88 TACR3 (0.68) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL297932 0.86 TACR3 (0.57) TACR3TACR1TACR2CCR5PPARG
SCHEMBL3275834 0.84 TACR3 (0.69) TACR3TACR1TACR2UBE2MDCUN1D1
SCHEMBL296569 0.84 TACR3 (0.68) TACR3TACR1TACR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033995-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-03-19 WO disclosed