SCHEMBL8050411

SCHEMBL8050411

C[C@]12CC[C@]3(O)c4ccccc4CC[C@@H]3[C@@H]1CCC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.50
ESR2 Q92731 2/20 0.50
STS P08842 3/20 0.46
SRD5A1 P18405 1/20 0.44
HSD17B3 P37058 3/20 0.44
CYP19A1 P11511 8/20 0.43
HSD17B1 P14061 3/20 0.43
CYP3A4 P08684 2/20 0.43
AKR1B10 O60218 1/20 0.43
LMNA P02545 1/20 0.43
SHBG P04278 1/20 0.43
CYP1A2 P05177 1/20 0.43
PGR P06401 1/20 0.43
SERPINA6 P08185 1/20 0.43
AR P10275 1/20 0.43
MAPT P10636 1/20 0.43
AKR1B1 P15121 1/20 0.43
NFKB1 P19838 1/20 0.43
SLC6A4 P31645 1/20 0.43
OPRM1 P35372 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13125425 0.84 ESR1 (0.57) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL15292941 0.84 ESR1 (0.57) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL11758322 0.84 ESR1 (0.57) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL1688725 0.83 ESR1 (0.71) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL11222251 0.80 STS (0.60) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL11671496 0.80 STS (0.60) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL8048295 0.80 STS (0.60) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL15295783 0.78 STS (0.57) ESR1ESR2STSCYP19A1HSD17B1
SCHEMBL8048190 0.77 SHBG (0.40) SRD5A1SHBG
SCHEMBL8038167 0.77 SHBG (0.40) SRD5A1SHBG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882735-B1 9 Alpha-hydroxy-8 alpha-estra-1,3,5(10)-trienes and a process for their preparation JENAPHARM GMBH (DE) 2000-04-19 EP disclosed
EP-0882735-A1 9 Alpha-hydroxy-8 alpha-estra-1,3,5(10)-trienes and a process for their preparation Jenapharm GmbH & Co. KG (DE) 1998-12-09 EP disclosed