SCHEMBL8050601

SCHEMBL8050601

Oc1cccc2nc(N3CCOCC3)sc12

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.61
NPC1 O15118 5/20 0.61
RAB9A P51151 5/20 0.61
AR P10275 5/20 0.56
ALOX15 P16050 2/20 0.51
GAA P10253 4/20 0.49
MAPT P10636 3/20 0.49
TP53 P04637 2/20 0.47
USP2 O75604 2/20 0.47
PKM P14618 1/20 0.47
POLB P06746 1/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 2/20 0.46
TSHR P16473 2/20 0.46
HSD17B10 Q99714 1/20 0.46
HTT P42858 1/20 0.44
ALOX5 P09917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3284981 0.84 SMN1; SMN2 (0.60) SMN1; SMN2NPC1RAB9AARALOX15
SCHEMBL3468625 0.82 KMT2A (0.45) SMN1; SMN2NPC1RAB9AMAPTPOLB
SCHEMBL20767964 0.82 SCN4A (0.46) SMN1; SMN2NPC1RAB9AUSP2ALDH1A1
SCHEMBL8057526 0.81 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9AARALOX15
SCHEMBL3287757 0.78 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9AARALOX15
SCHEMBL809829 0.76 RAB9A (1.00) SMN1; SMN2NPC1RAB9AARALOX15
SCHEMBL2096693 0.76 CHEK2 (0.46) SMN1; SMN2NPC1RAB9AGAAMAPT
SCHEMBL3284300 0.75 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AARALOX15
Hydrogen Sulfide SCHEMBL11606123 0.75 RAB9A (0.97) SMN1; SMN2NPC1RAB9AARALOX15
SCHEMBL5767716 0.74 SMN1; SMN2 (0.59) SMN1; SMN2NPC1RAB9AARALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed