SCHEMBL8051909

SCHEMBL8051909

CCc1ccccc1-n1c(Sc2ncc(S(C)(=O)=O)s2)nnc1-c1cccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 8/20 0.42
ALDH1A1 P00352 6/20 0.40
HSD17B10 Q99714 5/20 0.40
KDM4E B2RXH2 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
HPGD P15428 1/20 0.39
RECQL P46063 1/20 0.38
HTT P42858 2/20 0.38
LMNA P02545 1/20 0.38
APLNR P35414 3/20 0.38
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPK1 P28482 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042389 0.86 TSHR (0.57) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8044235 0.85 TSHR (0.43) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8041833 0.83 ALDH1A1 (0.46) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8050459 0.82 NPC1 (0.47) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8043091 0.82 TSHR (0.46) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8051552 0.82 KDM4E (0.53) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8047047 0.81 TSHR (0.52) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8042514 0.81 TSHR (0.46) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8717457 0.81 TSHR (0.41) TSHRALDH1A1HSD17B10KDM4ENPSR1
SCHEMBL8043939 0.81 TSHR (0.48) TSHRALDH1A1HSD17B10KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed