SCHEMBL8053095

SCHEMBL8053095

CCCCCCCCCCCCCCCCC(CN(O)C=O)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.50
GRIK2 Q13002 2/20 0.50
MAPT P10636 1/20 0.49
SLC1A2 P43004 1/20 0.47
SLC1A1 P43005 1/20 0.47
CA2 P00918 2/20 0.47
MAPK1 P28482 1/20 0.47
BMP1 P13497 2/20 0.46
GPR84 Q9NQS5 3/20 0.46
FFAR1 O14842 1/20 0.46
LCK P06239 1/20 0.44
PPARD Q03181 1/20 0.44
ZDHHC20 Q5W0Z9 1/20 0.44
ZDHHC2 Q9UIJ5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8053923 1.00 GRIK1 (0.50) GRIK1GRIK2MAPTSLC1A2SLC1A1
SCHEMBL4318257 0.98 GRIK1 (0.49) GRIK1GRIK2MAPTSLC1A2SLC1A1
SCHEMBL4956784 0.93 CA2 (0.55) SLC1A2SLC1A1CA2MAPK1BMP1
SCHEMBL3319613 0.93 CA2 (0.55) SLC1A2SLC1A1CA2MAPK1BMP1
SCHEMBL1191020 0.93 CA2 (0.55) SLC1A2SLC1A1CA2MAPK1BMP1
SCHEMBL3902711 0.83 CA2 (0.50) GRIK1GRIK2SLC1A2SLC1A1CA2
SCHEMBL3900866 0.83 CA2 (0.50) GRIK1GRIK2SLC1A2SLC1A1CA2
SCHEMBL25286591 0.78 GRIK1 (0.68) GRIK1GRIK2MAPTSLC1A2SLC1A1
SCHEMBL25295583 0.78 GRIK1 (0.68) GRIK1GRIK2MAPTSLC1A2SLC1A1
SCHEMBL25293243 0.78 GRIK1 (0.68) GRIK1GRIK2MAPTSLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028110-A Succinyl hydroxamic acid, N-formyl-N-hydroxy amino carboxylic acid and succinic acid amide derivatives as metalloprotease inhibitors BRITISH BIOTECH PHARMACEUTICALS LTD. (GB) 2000-02-22 US disclosed
EP-0763012-B1 SUCCINYL HYDROXAMIC ACID, N-FORMYL-N-HYDROXY AMINO CARBOXYLIC ACID AND SUCCINIC ACID AMIDE DERIVATIVES AS METALLOPROTEASE INHIBITORS BRITISH BIOTECH PHARM (GB) 1999-06-09 EP disclosed
EP-0763012-A1 SUCCINYL HYDROXAMIC ACID, N-FORMYL-N-HYDROXY AMINO CARBOXYLIC ACID AND SUCCINIC ACID AMIDE DERIVATIVES AS METALLOPROTEASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1997-03-19 EP disclosed
WO-1995032944-A1 SUCCINYL HYDROXAMIC ACID, N-FORMYL-N-HYDROXY AMINO CARBOXYLIC ACID AND SUCCINIC ACID AMIDE DERIVATIVES AS METALLOPROTEASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1995-12-07 WO disclosed