SCHEMBL8058565

SCHEMBL8058565

COc1ccccc1N1CCN(c2c(F)cc3c(=O)c(C(=O)O)cn(C4CC4)c3c2C(F)(F)F)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.52
ALDH1A1 P00352 6/20 0.52
KCNH2 Q12809 4/20 0.52
HPGD P15428 4/20 0.52
POLB P06746 3/20 0.52
TDP1 Q9NUW8 2/20 0.52
OPRM1 P35372 2/20 0.52
HSD17B10 Q99714 2/20 0.52
PRKD3 O94806 1/20 0.52
ALOX15 P16050 1/20 0.52
CLK2 P49760 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
LMNA P02545 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CYP2C19 P33261 1/20 0.49
GSK3B P49841 1/20 0.49
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
OPRD1 P41143 1/20 0.47
DPP4 P27487 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8057309 0.88 KDM4E (0.46) KDM4EALDH1A1HPGDPOLBHSD17B10
SCHEMBL8046825 0.87 KDM4E (0.54) KDM4EALDH1A1HPGDPOLBTDP1
SCHEMBL8061803 0.86 ALDH1A1 (0.53) KDM4EALDH1A1KCNH2HPGDPOLB
SCHEMBL8064182 0.86 KDM4E (0.45) KDM4EALDH1A1KCNH2HPGDPOLB
SCHEMBL8880183 0.85 KCNH2 (0.57) KDM4EALDH1A1KCNH2HPGDPOLB
SCHEMBL8061917 0.85 KDM4E (0.58) KDM4EALDH1A1HPGDPOLBTDP1
Hydrochloric Acid SCHEMBL8732413 0.85 KCNH2 (0.56) KDM4EALDH1A1KCNH2HPGDPOLB
SCHEMBL10401157 0.84 KDM4E (0.59) KDM4EALDH1A1KCNH2HPGDPOLB
SCHEMBL8064228 0.84 ALDH1A1 (0.52) KDM4EALDH1A1KCNH2HPGDPOLB
SCHEMBL27513354 0.82 ALDH1A1 (0.55) KDM4EALDH1A1KCNH2HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6034086-A VIRICIDES; AIDS THERAPY UBE INDUSTRIES, LTD. 2000-03-07 US disclosed
CN-1214632-A Remedies or preventives for AIDS SANKYO CO (JP) 1999-04-21 CN disclosed
EP-0878194-A1 REMEDIES OR PREVENTIVES FOR AIDS SANKYO COMPANY LIMITED (JP) 1998-11-18 EP disclosed
CN-1152916-A Trifluoromethylquinoline carboxylic acid derivative UBE INDUSTRIES (JP) 1997-06-25 CN disclosed
EP-0773214-A1 TRIFLUOROMETHYLQUINOLINECARBOXYLIC ACID DERIVATIVE UBE INDUSTRIES, LTD. (JP) 1997-05-14 EP disclosed