SCHEMBL8058744

SCHEMBL8058744

CC(C)(C#N)c1cc(C#N)cc(Cn2ccnc2)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 9/20 0.56
CYP19A1 P11511 7/20 0.56
CYP11B2 P19099 5/20 0.56
UGT1A4 P22310 1/20 0.49
PDE4D Q08499 1/20 0.49
FNTA P49354 3/20 0.43
FNTB P49356 3/20 0.43
PGGT1B P53609 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2350295 0.91 CYP19A1 (0.58) CYP11B1CYP19A1CYP11B2UGT1A4PDE4D
Anastrozole SCHEMBL9717292 0.81 CYP19A1 (0.79) CYP11B1CYP19A1CYP11B2UGT1A4PDE4D
SCHEMBL8070045 0.81 CYP11B1 (0.61) CYP11B1CYP19A1CYP11B2FNTAFNTB
SCHEMBL8074623 0.80 CYP19A1 (0.44) CYP11B1CYP19A1CYP11B2UGT1A4PDE4D
SCHEMBL8070226 0.79 CYP19A1 (0.50) CYP11B1CYP19A1CYP11B2FNTAFNTB
SCHEMBL13590044 0.79 CYP19A1 (0.68) CYP11B1CYP19A1CYP11B2UGT1A4PDE4D
SCHEMBL8059020 0.77 CYP19A1 (0.82) CYP19A1UGT1A4PDE4D
SCHEMBL14200258 0.74 CYP11B1 (0.62) CYP11B1CYP19A1CYP11B2
SCHEMBL17407556 0.74 CYP11B1 (0.62) CYP11B1CYP19A1CYP11B2
SCHEMBL4929247 0.73 CYP19A1 (0.60) CYP11B1CYP19A1CYP11B2UGT1A4PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36617-E Anastrozole and salts as anticancer agent ZENECA LIMITED (GB) 2000-03-14 US disclosed
EP-0296749-B1 (Substituted aralkyl) heterocyclic compounds ZENECA LTD (GB) 1994-10-26 EP disclosed
US-4935437-A (Substituted aralkyl) heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-19 US disclosed