SCHEMBL8070045

SCHEMBL8070045

CC(C)(C#N)c1cccc(Cn2ccnc2)c1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 11/20 0.61
CYP11B2 P19099 10/20 0.61
CYP19A1 P11511 5/20 0.61
ADRA2C P18825 1/20 0.55
FNTA P49354 3/20 0.54
FNTB P49356 3/20 0.54
PGGT1B P53609 3/20 0.54
CYP1A2 P05177 1/20 0.51
POLB P06746 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
MAPT P10636 1/20 0.51
TBXAS1 P24557 1/20 0.51
QPCT Q16769 1/20 0.51
CYP4Z1 Q86W10 1/20 0.51
QPCTL Q9NXS2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2350295 0.86 CYP19A1 (0.58) CYP11B1CYP11B2CYP19A1FNTAFNTB
SCHEMBL12245400 0.85 CYP11B1 (0.66) CYP11B1CYP11B2CYP19A1ADRA2CFNTA
SCHEMBL8058744 0.81 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1FNTAFNTB
SCHEMBL9747476 0.79 CYP11B1 (0.66) CYP11B1CYP11B2CYP19A1ADRA2CCYP1A2
SCHEMBL394308 0.78 CYP11B1 (0.83) CYP11B1CYP11B2CYP19A1ADRA2CCYP1A2
SCHEMBL13590044 0.77 CYP19A1 (0.68) CYP11B1CYP11B2CYP19A1TBXAS1
SCHEMBL12299569 0.77 CYP11B1 (0.71) CYP11B1CYP11B2CYP19A1ADRA2CCYP1A2
SCHEMBL8068082 0.77 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1ADRA2CCYP1A2
Anastrozole SCHEMBL9717292 0.77 CYP19A1 (0.79) CYP11B1CYP11B2CYP19A1
SCHEMBL24732609 0.76 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1ADRA2CFNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36617-E Anastrozole and salts as anticancer agent ZENECA LIMITED (GB) 2000-03-14 US disclosed
EP-0296749-B1 (Substituted aralkyl) heterocyclic compounds ZENECA LTD (GB) 1994-10-26 EP disclosed
US-4935437-A (Substituted aralkyl) heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-19 US disclosed