SCHEMBL8059441

SCHEMBL8059441

COC1CCc2c(C(=O)NC(=N)N)[nH]c3cccc1c23

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.39
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
DRD2 P14416 3/20 0.32
HTR1A P08908 2/20 0.32
MTNR1A P48039 3/20 0.32
MTNR1B P49286 3/20 0.32
MAPKAPK2 P49137 1/20 0.31
ACHE P22303 1/20 0.31
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
HTR5A P47898 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059448 0.96 PARP1 (0.36) PARP1ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL8070430 0.88 PARP1 (0.36) PARP1ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL8070427 0.82 PARP1 (0.38) PARP1ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL8059445 0.81 PARP1 (0.37) PARP1ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL8069957 0.81 PARP1 (0.38) PARP1ALDH1A1KDM4EMAPTDRD2
SCHEMBL8059450 0.79 PARP1 (0.36) PARP1ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL8069997 0.75 KDM4E (0.32) ALDH1A1KDM4EHSD17B10HPGDACHE
SCHEMBL8070000 0.73 PARP1 (0.50) PARP1ALDH1A1KDM4EMAPTDRD2
SCHEMBL8069950 0.72 MCL1 (0.40) PARP1ALDH1A1KDM4EMAPTHPGD
SCHEMBL8068495 0.71 PARP1 (0.38) PARP1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0803501-B1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMA (JP) 2000-07-05 EP disclosed
EP-0803501-A1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-29 EP disclosed