SCHEMBL8070000

SCHEMBL8070000

N=C(N)NC(=O)c1[nH]c2cccc3c2c1CCC3=O

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.50
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8073391 0.94 PARP1 (0.48) PARP1DRD2DRD1ALDH1A1KDM4E
SCHEMBL8059339 0.88 PARP1 (0.47) PARP1DRD2DRD1ALDH1A1KDM4E
SCHEMBL8070004 0.79 PARP1 (0.48) PARP1DRD2DRD1ALDH1A1KDM4E
SCHEMBL8068495 0.76 PARP1 (0.38) PARP1ALDH1A1KDM4EMAPT
SCHEMBL8073394 0.75 PARP1 (0.47) PARP1DRD2DRD1ALDH1A1KDM4E
SCHEMBL8069957 0.74 PARP1 (0.38) PARP1DRD2ALDH1A1KDM4EMAPT
SCHEMBL8069950 0.74 MCL1 (0.40) PARP1ALDH1A1KDM4EMAPT
SCHEMBL8059441 0.73 PARP1 (0.39) PARP1DRD2ALDH1A1KDM4EMAPT
SCHEMBL8068330 0.72 PARP1 (0.38) PARP1ALDH1A1KDM4EMAPT
SCHEMBL8070427 0.72 PARP1 (0.38) PARP1DRD2ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0803501-B1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMA (JP) 2000-07-05 EP disclosed
EP-0803501-A1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-29 EP disclosed