SCHEMBL8059974

SCHEMBL8059974

CC(N)Oc1cccc(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OGG1 O15527 1/20 0.58
GRM5 P41594 1/20 0.50
PNMT P11086 1/20 0.48
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SLC6A4 P31645 2/20 0.45
WDR5 P61964 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
HTR2A P28223 2/20 0.42
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
HTR7 P34969 1/20 0.42
HTR6 P50406 1/20 0.42
MAOB P27338 1/20 0.41
AOC3 Q16853 1/20 0.41
KCNH2 Q12809 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651909 0.85 TAAR1 (0.44) OGG1KMT2AALDH1A1MAPTHTR2A
SCHEMBL21394757 0.85 OGG1 (0.55) OGG1GRM5PNMTKMT2AL3MBTL1
Hydrazine SCHEMBL28120133 0.84 OGG1 (0.58) OGG1GRM5PNMTKMT2AL3MBTL1
SCHEMBL105734 0.83 OGG1 (0.57) OGG1GRM5KMT2AL3MBTL1SLC6A4
Chloromethane SCHEMBL27541396 0.82 OGG1 (0.56) OGG1GRM5KMT2AL3MBTL1SLC6A4
SCHEMBL10451483 0.82 OGG1 (0.56) OGG1GRM5PNMTKMT2AL3MBTL1
SCHEMBL10359842 0.80 OGG1 (0.58) OGG1GRM5KMT2AL3MBTL1SLC6A4
SCHEMBL17032600 0.80 OGG1 (0.54) OGG1GRM5PNMTKMT2AL3MBTL1
SCHEMBL11335792 0.80 OGG1 (0.54) OGG1GRM5PNMTKMT2AL3MBTL1
SCHEMBL3160383 0.80 OGG1 (0.54) OGG1GRM5PNMTKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3433234-B1 ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS MERCK SHARP & DOHME (US) 2021-10-27 EP disclosed
WO-2000012522-A1 MACROLIDE LHRH ANTAGONISTS ABBOTT LABORATORIES (US) 2000-03-09 WO disclosed
US-6020521-A Macrolide LHRH antagonists ABBOTT LABORATORIES (US) 2000-02-01 US disclosed
US-4119729-A TREATMENT OF HYPERTENSION MEAD JOHNSON & COMPANY (US) 1978-10-10 US disclosed
US-4067904-A ANTIARRHYTHMIA, HYPOTENSIVE MEAD JOHNSON & COMPANY (US) 1978-01-10 US disclosed