SCHEMBL8060729

SCHEMBL8060729

COC(=O)c1ccc2c(c1)S(=O)(=O)CNC2=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 1/20 0.44
KMT2A Q03164 2/20 0.43
CTDSP1 Q9GZU7 1/20 0.43
CA12 O43570 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
CA7 P43166 1/20 0.42
XDH P47989 1/20 0.42
CA14 Q9ULX7 1/20 0.42
ALDH1A1 P00352 6/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
ATM Q13315 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
LMNA P02545 2/20 0.41
CREBBP Q92793 1/20 0.40
CASP3 P42574 1/20 0.40
SLC40A1 Q9NP59 1/20 0.40
PDK2 Q15119 1/20 0.40
KDM4E B2RXH2 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058115 0.82 MAPT (0.39) CA12CA2CA9CA1CA7
SCHEMBL8058208 0.79 ALDH1A1 (0.49) KMT2ACA12CA2CA9CA1
SCHEMBL5904274 0.79 PTPRC (0.47) PTPRCKMT2ACA12CA2CA9
SCHEMBL8045078 0.77 MAPT (0.35) KMT2AALDH1A1ATMLMNAKDM4E
SCHEMBL1102209 0.77 ALDH1A1 (0.45) PTPRCKMT2ACA12CA2CA9
SCHEMBL8258364 0.76 CA1 (0.45) PTPRCKMT2ACA12CA2CA9
SCHEMBL31098601 0.76 SMYD3 (0.53) PTPRCKMT2ACTDSP1CA12CA2
SCHEMBL4611577 0.76 SMYD3 (0.53) PTPRCKMT2ACTDSP1CA12CA2
SCHEMBL22011240 0.75 KMT2A (0.47) PTPRCKMT2ACTDSP1CA12CA2
SCHEMBL22011243 0.75 KMT2A (0.47) PTPRCKMT2ACTDSP1CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed