SCHEMBL8060743

SCHEMBL8060743

COC(=O)c1ccc2c(c1)S(=O)(=O)C=CC2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA12 O43570 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
XDH P47989 1/20 0.42
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
HPGD P15428 4/20 0.40
MAPT P10636 4/20 0.40
HSD17B10 Q99714 3/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
ATM Q13315 1/20 0.40
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056319 0.80 ALDH1A1 (0.35) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8056207 0.75 TSHR (0.33) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8062794 0.72 CA1 (0.44) CA1CA2CA12CA7CA9
SCHEMBL8062954 0.70 ALDH1A1 (0.44) CA1CA2CA12CA7CA9
SCHEMBL1574104 0.69 PTPRC (0.49) CA1CA2CA12CA7CA9
SCHEMBL8060718 0.69 CA12 (0.44) CA1CA2CA12CA7CA9
SCHEMBL8045056 0.69 CA1 (0.44) CA1CA2CA12CA7CA9
SCHEMBL8045295 0.69 CA12 (0.41) CA1CA2CA12CA7CA9
SCHEMBL18682115 0.69 CA1 (0.55) CA1CA2CA12CA7CA9
SCHEMBL18670723 0.69 CA1 (0.55) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed