SCHEMBL806116

SCHEMBL806116

Cn1c(C(=O)NCC2CC2)nc2c(N3CCC(N)(c4ccccc4)CC3)ncnc21

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.60
PIK3R1 P27986 1/20 0.60
CNR1 P21554 12/20 0.43
CNR2 P34972 10/20 0.43
AKT1 P31749 2/20 0.40
AKT2 P31751 2/20 0.40
NAPEPLD Q6IQ20 1/20 0.36
MAP4K4 O95819 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL787665 0.90 PIK3CD (0.61) PIK3CDPIK3R1CNR1CNR2NAPEPLD
SCHEMBL788059 0.87 PIK3CD (0.58) PIK3CDPIK3R1CNR1CNR2
SCHEMBL806202 0.84 PIK3CD (0.66) PIK3CDPIK3R1CNR1CNR2NAPEPLD
SCHEMBL794109 0.83 PIK3CD (0.59) PIK3CDPIK3R1CNR1CNR2NAPEPLD
SCHEMBL806199 0.82 PIK3CD (0.60) PIK3CDPIK3R1CNR1CNR2
SCHEMBL806198 0.82 PIK3CD (0.60) PIK3CDPIK3R1CNR1CNR2
SCHEMBL788072 0.82 PIK3CD (0.58) PIK3CDPIK3R1CNR1CNR2NAPEPLD
SCHEMBL18175791 0.82 PIK3CD (0.63) PIK3CDPIK3R1CNR1CNR2
SCHEMBL806241 0.81 PIK3CD (0.57) PIK3CDPIK3R1
SCHEMBL788225 0.81 PIK3CD (0.56) PIK3CDPIK3R1CNR1CNR2NAPEPLD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037226-A1 INHIBITORS OF PI3K-DELTA AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-03-22 WO disclosed