SCHEMBL8062874

SCHEMBL8062874

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)C=C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 4/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
ALDH1A1 P00352 10/20 0.35
KDM4E B2RXH2 9/20 0.35
MAPT P10636 4/20 0.35
HSD17B10 Q99714 4/20 0.35
HTT P42858 1/20 0.35
CA12 O43570 1/20 0.34
HPGD P15428 4/20 0.34
LMNA P02545 3/20 0.34
GAA P10253 2/20 0.33
GLA P06280 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
ATM Q13315 1/20 0.33
PLCG2 P16885 1/20 0.33
KMT2A Q03164 3/20 0.33
NR4A2 P43354 1/20 0.32
CFTR P13569 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056963 0.82 KDM4E (0.38) CA9CA1CA2ALDH1A1KDM4E
SCHEMBL8056361 0.79 ALDH1A1 (0.33) ALDH1A1KDM4EMAPTHSD17B10HTT
SCHEMBL8057300 0.78 CFTR (0.46) CA9CA1CA2ALDH1A1KDM4E
SCHEMBL8056470 0.78 ALDH1A1 (0.34) ALDH1A1KDM4EMAPTHSD17B10HTT
SCHEMBL8057086 0.78 ALDH1A1 (0.32) CA9CA1CA2ALDH1A1KDM4E
SCHEMBL8060886 0.76 ALDH1A1 (0.33) ALDH1A1KDM4EMAPTHSD17B10HTT
SCHEMBL8057109 0.75 ALDH1A1 (0.34) CA9CA1CA2ALDH1A1KDM4E
SCHEMBL8056207 0.75 TSHR (0.33) ALDH1A1KDM4EMAPTHSD17B10HTT
SCHEMBL8058137 0.72 ALDH1A1 (0.36) CA9CA1CA2ALDH1A1KDM4E
SCHEMBL8060681 0.72 ALDH1A1 (0.32) ALDH1A1KDM4EMAPTHSD17B10HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed