SCHEMBL8062894

SCHEMBL8062894

COC(=O)c1cc2c(cc1C(F)(F)F)C(=O)CS2(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CFTR P13569 6/20 0.40
NOTUM Q6P988 2/20 0.39
VEGFA P15692 1/20 0.36
MAPT P10636 1/20 0.35
KCNN4 O15554 2/20 0.33
SOS1 Q07889 1/20 0.33
ESRRA P11474 1/20 0.33
PDK2 Q15119 3/20 0.33
P4HB P07237 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056417 0.86 CFTR (0.39) CFTRNOTUMMAPTKCNN4SOS1
SCHEMBL8056235 0.84 CFTR (0.38) CFTRNOTUMMAPTKCNN4SOS1
SCHEMBL8056232 0.84 CFTR (0.38) CFTRNOTUMMAPTKCNN4SOS1
SCHEMBL8058223 0.83 CFTR (0.37) CFTRNOTUMMAPTKCNN4SOS1
SCHEMBL8058221 0.83 CFTR (0.37) CFTRNOTUMMAPTKCNN4SOS1
SCHEMBL8058193 0.82 VEGFA (0.41) VEGFAMAPTKCNN4PDK2
SCHEMBL8057061 0.81 KDM4E (0.36) VEGFAMAPT
SCHEMBL8045172 0.78 VEGFA (0.35) VEGFAMAPT
SCHEMBL8056401 0.77
SCHEMBL8062790 0.75 NOTUM (0.43) CFTRNOTUMMAPTSOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed