SCHEMBL8064263

SCHEMBL8064263

COc1cc(C)c(S(=O)(=O)OC(=O)[C@@H](N)CCCNC(=N)N)c(C)c1C

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 5/20 0.40
F2 P00734 1/20 0.39
AVPR1A P37288 4/20 0.38
PLG P00747 1/20 0.35
NPY4R P50391 2/20 0.35
NPY1R P25929 1/20 0.35
EPHX2 P34913 1/20 0.34
NMT1 P30419 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MARS1 P56192 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30038580 0.80 AVPR1B (0.43) AVPR1BF2AVPR1APLGNMT1
SCHEMBL24136539 0.80 AVPR1B (0.43) AVPR1BF2AVPR1APLGNMT1
SCHEMBL22139318 0.80 AVPR1B (0.43) AVPR1BF2AVPR1APLGNMT1
SCHEMBL9329697 0.79 AVPR1B (0.52) AVPR1BF2AVPR1APLG
SCHEMBL4901697 0.78 AVPR1B (0.42) AVPR1BF2AVPR1APLGNMT1
SCHEMBL7898282 0.78 AVPR1B (0.54) AVPR1BF2AVPR1APLG
SCHEMBL1509780 0.78 AVPR1B (0.54) AVPR1BF2AVPR1APLG
SCHEMBL30007346 0.78 AVPR1B (0.54) AVPR1BF2AVPR1APLG
SCHEMBL1509781 0.78 AVPR1B (0.54) AVPR1BF2AVPR1APLG
Hydrochloric Acid SCHEMBL4901689 0.78 AVPR1B (0.42) AVPR1BF2AVPR1APLGNMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643778-B1 ENCODED COMBINATORIAL CHEMICAL LIBRARIES SCRIPPS RESEARCH INST (US) 2000-05-31 EP disclosed
EP-0643778-A4 ENCODED COMBINATORIAL CHEMICAL LIBRARIES. SCRIPPS RESEARCH INST (US) 1995-09-20 EP disclosed
EP-0643778-A1 ENCODED COMBINATORIAL CHEMICAL LIBRARIES THE SCRIPPS RESEARCH INSTITUTE (US) 1995-03-22 EP disclosed
WO-1993020242-A1 ENCODED COMBINATORIAL CHEMICAL LIBRARIES THE SCRIPPS RESEARCH INSTITUTE (US) 1993-10-14 WO disclosed