SCHEMBL8064347

SCHEMBL8064347

C[C@@H]1C[C@H](COCCCOc2ccccc2)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.42
HRH3 Q9Y5N1 4/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
GPR119 Q8TDV5 5/20 0.39
SRC P12931 4/20 0.38
NR1H2 P55055 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13663655 0.89 PDE4B (0.42) PDE4BNPC1HPGDRAB9AGPR119
SCHEMBL8064836 0.89 SRC (0.41) PDE4BSRCNR1H2
SCHEMBL3945721 0.88 PDE4B (0.42) PDE4BNPC1HPGDRAB9AGPR119
SCHEMBL13663724 0.83 PDE4B (0.39) PDE4BNPC1HPGDRAB9AGPR119
SCHEMBL4297046 0.83 ABCB1 (0.39) PDE4BNPC1HPGDRAB9AGPR119
SCHEMBL13765329 0.82 MEN1 (0.36) NR1H2
SCHEMBL8064390 0.78 HDAC8 (0.42)
SCHEMBL25694140 0.78 CHRNB2 (0.47) NPC1SRC
SCHEMBL8059551 0.78 CYP1A2 (0.45) PDE4BSRCNR1H2
SCHEMBL16080305 0.77 NR1H2 (0.51) SRCNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026197-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE GLAXO GROUP LIMITED (GB) 2009-02-26 WO disclosed