SCHEMBL8065026

SCHEMBL8065026

N[C@@H](Cc1ccccc1)C(=O)OC(=O)N1CCN(c2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.54
GFER P55789 1/20 0.54
HTT P42858 1/20 0.52
GRM5 P41594 1/20 0.49
ROCK2 O75116 1/20 0.47
CYP3A4 P08684 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 3/20 0.46
MAPT P10636 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
HDAC8 Q9BY41 2/20 0.46
LMNA P02545 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ALPI P09923 1/20 0.45
PKM P14618 1/20 0.45
PTGS1 P23219 1/20 0.45
XIAP P98170 1/20 0.45
SLC7A5 Q01650 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065024 0.90 POLB (0.54) POLBGFERHTTGRM5ROCK2
SCHEMBL8059247 0.87 HDAC8 (0.48) POLBALDH1A1HDAC8ALPIPKM
SCHEMBL10491053 0.86 KMT2A (0.59) POLBHTTKDM4EALDH1A1SMN1; SMN2
SCHEMBL11947653 0.82 POLB (0.54) POLBGFERHTTGRM5KDM4E
SCHEMBL31627496 0.81 MEN1 (0.53) POLBGFERGRM5KDM4EMAPT
SCHEMBL34468319 0.81 MEN1 (0.53) POLBGFERGRM5KDM4EMAPT
SCHEMBL288607 0.77 SLC7A5 (0.68) HDAC8ALPIPKMPTGS1XIAP
SCHEMBL8835936 0.77 SLC7A5 (0.68) HDAC8ALPIPKMPTGS1XIAP
SCHEMBL28820471 0.77 SLC7A5 (0.68) HDAC8ALPIPKMPTGS1XIAP
SCHEMBL9727540 0.76 NPSR1 (0.68) GRM5KDM4EMAPTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000051-A1 CARBAMYLOXY COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-17 EP disclosed
WO-1999006390-A1 CARBAMYLOXY COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed