SCHEMBL8065775

SCHEMBL8065775

COc1ccc(-c2ccc3cccc(CCNC(C)=O)c3c2)cc1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 20/20 0.82
MTNR1B P49286 13/20 0.82
HTR2C P28335 1/20 0.82
HTR2B P41595 1/20 0.82
NQO2 P16083 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8054339 0.92 MTNR1A (0.80) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL1158495 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL29930659 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL27844916 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL114476 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
SCHEMBL7016328 0.90 MTNR1A (1.00) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL28522576 0.89 MTNR1A (0.97) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL28116100 0.89 MTNR1A (0.97) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL1289524 0.89 MTNR1A (0.97) MTNR1AMTNR1BHTR2CHTR2BNQO2
Agomelatine SCHEMBL27785485 0.89 MTNR1A (0.97) MTNR1AMTNR1BHTR2CHTR2BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143789-A ENANTIOMORPHS ADIR ET COMPAGNIE (FR) 2000-11-07 US disclosed
EP-0919541-A1 Naphthalene compounds, process for their preparation and their pharmaceutical compositions ADIR ET COMPAGNIE (FR) 1999-06-02 EP disclosed