SCHEMBL8065832

SCHEMBL8065832

C[C@]12CCC(=O)N[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)[C@@H](Oc3ccc([N+](=O)[O-])cc3)CC[C@@H]12

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 4/20 0.49
SRD5A2 P31213 4/20 0.48
AR P10275 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065834 1.00 SRD5A1 (0.49) SRD5A1SRD5A2AR
SCHEMBL3278549 0.88 SRD5A2 (0.61) SRD5A1SRD5A2AR
SCHEMBL3276274 0.87 SRD5A1 (0.52) SRD5A1SRD5A2AR
SCHEMBL8075695 0.85 SRD5A1 (0.52) SRD5A1SRD5A2AR
SCHEMBL8075699 0.85 SRD5A1 (0.52) SRD5A1SRD5A2AR
SCHEMBL9003279 0.81 CYP19A1 (0.54) SRD5A2AR
SCHEMBL8073236 0.80 SRD5A1 (0.60) SRD5A1SRD5A2
SCHEMBL8073237 0.80 SRD5A1 (0.60) SRD5A1SRD5A2
SCHEMBL8712728 0.78 SRD5A1 (0.60) SRD5A1SRD5A2AR
SCHEMBL7611331 0.77 SRD5A1 (0.58) SRD5A1SRD5A2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641204-B1 17-ETHERS AND THIOETHERS OF 4-AZA-STEROIDS MERCK & CO INC (US) 2000-08-16 EP claimed
US-5536727-A TREATMENT OF HYPERANDROGENIC DISEASES MERCK & CO., INC. (US) 1996-07-16 US claimed
EP-0641204-A4 17-ETHERS AND THIOETHERS OF 4-AZA-STEROIDS. MERCK & CO INC (US) 1995-08-23 EP claimed
EP-0641204-A1 17-ETHERS AND THIOETHERS OF 4-AZA-STEROIDS MERCK & CO. INC. (US) 1995-03-08 EP claimed
WO-1993023040-A1 17-ETHERS AND THIOETHERS OF 4-AZA-STEROIDS MERCK & CO., INC. (US) 1993-11-25 WO claimed
EP-0641204-B1 17-ETHERS AND THIOETHERS OF 4-AZA-STEROIDS MERCK & CO INC (US) 2000-08-16 EP disclosed
WO-1993023040-A1 17-ETHERS AND THIOETHERS OF 4-AZA-STEROIDS MERCK & CO., INC. (US) 1993-11-25 WO disclosed