SCHEMBL8066586

SCHEMBL8066586

COC(=O)Cc1cccc([C@@H]2CN(C)Cc3ccccc32)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 20/20 0.55
SLC6A4 P31645 20/20 0.55
SLC6A3 Q01959 20/20 0.55
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8066583 1.00 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8057428 0.87 SLC6A2 (0.63) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8057430 0.86 SLC6A2 (0.58) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8057433 0.86 SLC6A2 (0.58) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8057198 0.79 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8068783 0.79 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3
SCHEMBL8057082 0.76 SLC6A2 (0.56) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8057194 0.74 SLC6A2 (0.68) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8057196 0.74 SLC6A2 (0.68) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL4032379 0.73 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028080-A Quinolin-2-(1H)-ones MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-02-22 US disclosed