SCHEMBL8067334

SCHEMBL8067334

CS(=O)(=O)N1CC2(CCN(C(=O)OCc3ccccc3)CC2)c2cc(F)ccc21

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.57
NPY5R Q15761 1/20 0.51
GHSR Q92847 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29661999 1.00 TACR1 (0.57) TACR1NPY5RGHSR
SCHEMBL29661957 0.89 RORC (0.46) TACR1
SCHEMBL2878354 0.88 TACR1 (0.68) TACR1NPY5RGHSR
SCHEMBL2625791 0.87 HDAC1 (0.50) TACR1
SCHEMBL4974614 0.87 HDAC1 (0.50) TACR1
SCHEMBL29662002 0.86 TACR1 (0.50) TACR1NPY5RGHSR
SCHEMBL2632889 0.85 HDAC1 (0.54) TACR1
SCHEMBL26969702 0.84 GNRHR (0.47) TACR1
SCHEMBL13180673 0.81 HDAC1 (0.45) TACR1
SCHEMBL20955202 0.81 XIAP (0.46) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013652-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIHISTAMINES MERCK & CO., INC. (US) 2000-01-11 US disclosed
US-5962462-A COMPOUNDS WHICH INHIBIT THE ENTRY OF HUMAN IMMUNODEFICIENCY VIRUS (HIV) INTO TARGET CELLS; DELAYING THE ONSET OF ACQUIRED IMMUNE DEFICIENCY SYNDROME (AIDS). MERCK & CO., INC. (US) 1999-10-05 US disclosed