SCHEMBL806853

SCHEMBL806853

CCCn1c(Cl)nc2nc(-c3cnn(Cc4cccc(CF)c4)c3)n(COC(=O)C(C)(C)C)c2c1=O

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 20/20 0.41
ADORA1 P30542 17/20 0.41
ADORA2A P29274 16/20 0.41
ADORA3 P0DMS8 11/20 0.40
PLK4 O00444 1/20 0.38
CDK2 P24941 1/20 0.38
IRAK1 P51617 1/20 0.38
RPS6KA3 P51812 1/20 0.38
PLK3 Q9H4B4 1/20 0.38
CSNK1G3 Q9Y6M4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18133300 0.94 ADORA2B (0.42) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL15064882 0.91 ADORA2B (0.50) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL796991 0.83 ADORA2B (0.50) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL18133294 0.82 ADORA2B (0.46) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL15064746 0.81 ADORA2B (0.48) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL15064429 0.81 ADORA2B (0.54) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL15064477 0.81 ADORA2B (0.48) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL30891831 0.80 ADORA2B (0.47) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL797120 0.80 ADORA2B (0.47) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL30891869 0.79 ADORA2B (0.51) ADORA2BADORA1ADORA2AADORA3PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035548-A1 PURINE COMPOUNDS AS PRODRUGS OF A2B ADENOSINE RECEPTOR ANTAGONISTS, THEIR PROCESS AND MEDICINAL APPLICATIONS ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2012-03-22 WO disclosed