SCHEMBL806883

SCHEMBL806883

Cc1ccc(CCC(=O)N2CCC3(CC2)CN/C(=N\C(=O)c2nc(Cl)c(N)nc2N)N3)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
GPBAR1 Q8TDU6 1/20 0.34
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
ENPP2 Q13822 3/20 0.34
ATXN2 Q99700 2/20 0.34
SCNN1A P37088 5/20 0.33
DGAT1 O75907 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1684500 0.93 SCNN1A (0.35) ALDH1A1ENPP2ATXN2SCNN1A
SCHEMBL1684511 0.93 SCNN1A (0.35) ALDH1A1ENPP2ATXN2SCNN1A
SCHEMBL1684543 0.93 SCNN1A (0.41) ALDH1A1ENPP2ATXN2SCNN1A
SCHEMBL1684608 0.92 ALDH1A1 (0.42) ALDH1A1KMT2AMEN1ENPP2ATXN2
SCHEMBL1684603 0.92 ALDH1A1 (0.42) ALDH1A1KMT2AMEN1ENPP2ATXN2
SCHEMBL1684527 0.91 ALDH1A1 (0.44) ALDH1A1GPBAR1KMT2AMEN1SCNN1A
SCHEMBL1587241 0.91 SCNN1A (0.36) ALDH1A1KMT2AMEN1ENPP2ATXN2
SCHEMBL1587243 0.91 SCNN1A (0.36) ALDH1A1KMT2AMEN1ENPP2ATXN2
SCHEMBL19392998 0.90 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1ENPP2ATXN2
SCHEMBL1684842 0.89 ALDH1A1 (0.38) ALDH1A1KMT2AMEN1ENPP2ATXN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035158-A1 PYRAZINE DERIVATIVES AS ENAC BLOCKERS NOVARTIS AG (CH) 2012-03-22 WO disclosed