SCHEMBL8069736

SCHEMBL8069736

BCc1ccc(OC)c(-c2cccc(Cl)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 7/20 0.60
PDE4D Q08499 2/20 0.58
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALOX5 P09917 1/20 0.42
GABRA1 P14867 1/20 0.42
CNR2 P34972 1/20 0.42
GABRB2 P47870 1/20 0.42
TAAR1 Q96RJ0 2/20 0.41
PTGES2 Q9H7Z7 1/20 0.41
MAPK10 P53779 1/20 0.41
HTR7 P34969 2/20 0.41
RORC P51449 1/20 0.41
RORB Q92753 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28709947 0.87 PDE4B (0.62) PDE4BPDE4DNPC1MAPTTSHR
SCHEMBL13578468 0.85 PDE4D (0.61) PDE4BPDE4DNPC1MAPTTSHR
SCHEMBL29406552 0.85 PDE4D (0.61) PDE4BPDE4DNPC1MAPTTSHR
SCHEMBL3466479 0.85 PDE4B (0.60) PDE4BPDE4DNPC1MAPTTSHR
SCHEMBL5099550 0.82 PDE4D (0.56) PDE4BPDE4DNPC1MAPTTSHR
SCHEMBL8063138 0.82 PDE4B (0.63) PDE4BPDE4DTAAR1
Hydrochloric Acid SCHEMBL3793938 0.81 PDE4D (0.69) PDE4BPDE4DTAAR1PTGES2MAPK10
SCHEMBL3788487 0.81 PDE4D (0.69) PDE4BPDE4DTAAR1PTGES2MAPK10
SCHEMBL17633592 0.81 PDE4D (0.66) PDE4BPDE4DSMN1; SMN2MAPK10HTR7
SCHEMBL8065449 0.81 PDE4D (0.63) PDE4BPDE4DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067600-A2 BIARYL PDE4 INHIBITORS FOR TREATING INFLAMMATION DECODE GENETICS EHF (IS) 2009-05-28 WO disclosed