SCHEMBL807047

SCHEMBL807047

Nc1nc2ccc(Cl)cc2cc1-c1cn[nH]c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.44
ROCK2 O75116 6/20 0.41
ROCK1 Q13464 3/20 0.39
AKT2 P31751 5/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
NOS1 P29475 1/20 0.38
AKT1 P31749 3/20 0.38
PRKACA P17612 2/20 0.37
AKT3 Q9Y243 2/20 0.37
RPS6KA5 O75582 1/20 0.37
RPS6KA4 O75676 1/20 0.37
LATS1 O95835 1/20 0.37
PRKACB P22694 1/20 0.37
RPS6KB1 P23443 1/20 0.37
GRK2 P25098 1/20 0.37
RPS6KA3 P51812 1/20 0.37
PRKCD Q05655 1/20 0.37
RPS6KA2 Q15349 1/20 0.37
RPS6KA1 Q15418 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26613585 0.75 KCNH2 (0.46) ROCK2ROCK1AKT2NOS1AKT1
SCHEMBL29746235 0.75 KCNH2 (0.46) ROCK2ROCK1AKT2NOS1AKT1
SCHEMBL24802714 0.72 TDP1 (0.44) ROCK2ROCK1AKT2
SCHEMBL19398632 0.72 AHR (0.50) ROCK2ROCK1AKT2AKT1PRKACA
SCHEMBL790083 0.70 PTGS2 (0.51)
SCHEMBL7262530 0.70 PIK3CG (0.47) PDE3A
SCHEMBL21405437 0.69 LRRK2 (0.47) LRRK2ROCK2ROCK1AKT2AKT1
SCHEMBL16983118 0.69 PDE3B (0.49) LRRK2ROCK2ROCK1PDE3BPDE3A
SCHEMBL790542 0.69 SRC (0.49) PIK3CA
SCHEMBL509823 0.68 LRRK2 (0.45) LRRK2ROCK2ROCK1AKT2AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed