SCHEMBL8070669

SCHEMBL8070669

COc1c(C)cnc(CSc2nc3cc(N4CCCCC4)c(F)cc3[nH]2)c1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 2/20 0.59
OPRL1 P41146 13/20 0.51
PDE10A Q9Y233 1/20 0.41
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
CYP2C9 P11712 2/20 0.37
WDR5 P61964 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
DDAH1 O94760 1/20 0.37
ABCB11 O95342 1/20 0.37
ATP1A1 P05023 1/20 0.37
ATP1B1 P05026 1/20 0.37
CYP1A2 P05177 1/20 0.37
CHRM2 P08172 1/20 0.37
ABCB1 P08183 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8061857 0.92 OPRL1 (0.60) BRS3OPRL1ALDH1A1TSHRCYP2C9
SCHEMBL8059921 0.85 BRS3 (0.51) BRS3OPRL1ALDH1A1TSHRKDM4E
SCHEMBL8075357 0.84 OPRL1 (0.53) BRS3OPRL1CYP2C9ATP1A1ATP1B1
SCHEMBL8060096 0.84 OPRL1 (0.53) BRS3OPRL1CYP2C9ATP1A1ATP1B1
SCHEMBL8071079 0.83 OPRL1 (0.58) BRS3OPRL1ALDH1A1TSHREGLN1
SCHEMBL8072215 0.83 OPRL1 (0.54) BRS3OPRL1CYP2C9ATP1A1ATP1B1
SCHEMBL8074070 0.82 BRS3 (0.58) BRS3OPRL1ALDH1A1CYP2C9WDR5
SCHEMBL8060015 0.81 PDE10A (0.40) BRS3OPRL1PDE10AALDH1A1EGLN1
SCHEMBL8070545 0.78 NPC1 (0.62) BRS3OPRL1ALDH1A1TSHRCYP2C9
SCHEMBL9784719 0.76 BRS3 (0.67) BRS3ALDH1A1CYP2C9WDR5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US claimed
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US disclosed
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed