SCHEMBL8074070

SCHEMBL8074070

COc1c(C)cnc(CSc2nc3cc(-n4ccnc4)c(F)cc3[nH]2)c1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 2/20 0.58
OPRL1 P41146 10/20 0.40
SHMT2 P34897 1/20 0.37
CYP2C9 P11712 3/20 0.36
WDR5 P61964 3/20 0.36
KMT2A Q03164 3/20 0.36
ATP1A1 P05023 2/20 0.36
ATP1B1 P05026 2/20 0.36
ATP1A3 P13637 2/20 0.36
ATP1B2 P14415 2/20 0.36
ATP4A P20648 2/20 0.36
ATP1A2 P50993 2/20 0.36
ATP4B P51164 2/20 0.36
ATP1B3 P54709 2/20 0.36
FXYD2 P54710 2/20 0.36
ATP1A4 Q13733 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
HTT P42858 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071118 0.85 NPC1 (0.47) BRS3OPRL1CYP2C9ATP1A1ATP1B1
SCHEMBL8070669 0.82 BRS3 (0.59) BRS3OPRL1CYP2C9WDR5KMT2A
SCHEMBL8061857 0.82 OPRL1 (0.60) BRS3OPRL1SHMT2CYP2C9WDR5
SCHEMBL8070793 0.81 OPRL1 (0.44) BRS3OPRL1CYP2C9CYP1A2CYP3A4
SCHEMBL8071182 0.81 OPRL1 (0.44) OPRL1CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL8074080 0.81 CYP2C9 (0.59) BRS3OPRL1CYP2C9WDR5KMT2A
SCHEMBL8059870 0.81 BRS3 (0.36) BRS3CYP2C9WDR5KMT2AATP1A1
SCHEMBL8070664 0.81 CYP2C9 (0.46) BRS3OPRL1CYP2C9WDR5KMT2A
SCHEMBL8059958 0.79 NPC1 (0.61) BRS3OPRL1CYP2C9WDR5KMT2A
SCHEMBL8071180 0.78 NOS2 (0.58) BRS3OPRL1CYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US claimed
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US disclosed
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed