SCHEMBL8070828

SCHEMBL8070828

CC(C)(C)OC(=O)N[C@@H](Cc1cccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)O)c1)C(=O)NCC(=O)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.59
CTSK P43235 8/20 0.59
CTSB P07858 7/20 0.59
CTSL P07711 5/20 0.57
ACE P12821 1/20 0.55
SYK P43405 1/20 0.51
PPARA Q07869 1/20 0.51
AKT1 P31749 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19837597 0.90 CTSS (0.69) CTSSCTSKCTSBCTSLPPARA
SCHEMBL18154315 0.90 CTSS (0.69) CTSSCTSKCTSBCTSLPPARA
SCHEMBL11123304 0.90 CTSS (0.69) CTSSCTSKCTSBCTSLPPARA
SCHEMBL8072132 0.87 ACE (0.60) CTSSCTSKCTSBCTSLACE
SCHEMBL8072127 0.87 ACE (0.60) CTSSCTSKCTSBCTSLACE
SCHEMBL10054705 0.86 ACE (0.59) CTSSCTSKCTSBCTSLACE
SCHEMBL10054782 0.86 ACE (0.59) CTSSCTSKCTSBCTSLACE
SCHEMBL30100566 0.84 CTSS (0.63) CTSSCTSKCTSBCTSLACE
SCHEMBL11120671 0.84 CTSS (0.66) CTSSCTSKCTSBCTSLAKT1
SCHEMBL30100571 0.84 CTSS (0.58) CTSSCTSKCTSBCTSLACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080838-A SYNTHETIC CONSTRUCT PREPARED TO HOLD TWO PEPTIDE HELICES IN TIGHT ARRANGEMENT TO MIMIC DNA BINDING CONFORMATION; FOR INVESSTIGATIONAL STUDIES UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2000-06-27 US disclosed