SCHEMBL8074040

SCHEMBL8074040

CC(C)(C)OC(=O)N1CCN(c2cc3nc(S)[nH]c3cc2F)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTT P42858 2/20 0.47
NAMPT P43490 1/20 0.44
KCNH2 Q12809 1/20 0.43
OPRL1 P41146 3/20 0.42
GPR119 Q8TDV5 4/20 0.41
EGLN1 Q9GZT9 1/20 0.40
MAP4K4 O95819 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
KIT P10721 1/20 0.40
SMARCA2 P51531 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070660 0.82 OPRL1 (0.46) ALDH1A1MAPTKDM4EPOLBGAA
SCHEMBL23123045 0.82 ALDH1A1 (0.47) ALDH1A1MAPTKDM4EPOLBGAA
SCHEMBL8059756 0.81 MAPT (0.49) ALDH1A1MAPTTSHRNAMPTKCNH2
SCHEMBL8069092 0.79 OPRL1 (0.57) ALDH1A1MAPTOPRL1EGLN1
SCHEMBL6494859 0.78 MAPT (0.74) ALDH1A1MAPTKDM4EPOLBGAA
SCHEMBL21937028 0.78 MAPT (0.51) ALDH1A1MAPTKDM4EPOLBGAA
SCHEMBL8068945 0.77 OPRL1 (0.51) ALDH1A1ALOX15HSD17B10OPRL1EGLN1
SCHEMBL8071080 0.76 EGLN1 (0.52) HPGDTSHROPRL1EGLN1
SCHEMBL8070777 0.76 EGLN1 (0.52) HPGDTSHROPRL1EGLN1
SCHEMBL6486955 0.76 OPRL1 (0.48) NAMPTKCNH2OPRL1EGLN1MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US disclosed
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed