SCHEMBL8074175

SCHEMBL8074175

O=C1c2ccccc2C(=O)N1C1(F)CCCC1.O=C1c2ccccc2C(=O)N1C1(O)CCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.43
KDM4E B2RXH2 5/20 0.38
HPGD P15428 5/20 0.38
HSD17B10 Q99714 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
TSHR P16473 3/20 0.38
MAPK1 P28482 2/20 0.38
LMNA P02545 3/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ALOX12 P18054 2/20 0.33
CA9 Q16790 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CASP1 P29466 1/20 0.33
CA7 P43166 1/20 0.33
RECQL P46063 1/20 0.33
BACE1 P56817 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6662082 0.90 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL6659478 0.90 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL5502763 0.88 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL28664942 0.68 ALDH1A1 (0.68) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL5958862 0.68 TDP1 (0.35) ALDH1A1SMN1; SMN2TSHRCYP2C19PKM
SCHEMBL10806351 0.67 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL11360248 0.67 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL11728360 0.67 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL11611884 0.67 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL29885176 0.67 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027363-A2 ADENOSINE A1-RECEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 2000-08-16 EP disclosed
WO-1999024450-A2 ADENSINE A1 RECEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 1999-05-20 WO disclosed