SCHEMBL8074265

SCHEMBL8074265

COC(=O)[C@H]1CCc2c(cccc2OC)C1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.64
MTNR1B P49286 5/20 0.64
CA1 P00915 3/20 0.61
CA2 P00918 3/20 0.61
ACHE P22303 3/20 0.61
DRD2 P14416 9/20 0.59
DRD3 P35462 7/20 0.59
DRD4 P21917 5/20 0.59
CHRM2 P08172 1/20 0.55
CHRM1 P11229 1/20 0.55
CHRM3 P20309 1/20 0.55
CYP1A2 P05177 1/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALOX15 P16050 1/20 0.51
EPHX2 P34913 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6819517 1.00 MTNR1A (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL5835471 0.90 MTNR1A (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL8066344 0.90 MTNR1A (0.64) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL8080874 0.87 MTNR1A (0.61) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL8605995 0.87 MTNR1A (0.61) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL7778584 0.87 MTNR1A (0.61) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL8158536 0.85 MTNR1A (0.49) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL20096622 0.83 CYP1A2 (0.46) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL7924693 0.83 CYP1A2 (0.46) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL10983820 0.82 CYP1A2 (0.61) MTNR1AMTNR1BCA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683236-B1 Enzymatic process for the preparation of optical active tetralin-derivatives SANOFI SYNTHELABO (FR) 2000-08-09 EP claimed
EP-0683236-B1 Enzymatic process for the preparation of optical active tetralin-derivatives SANOFI SYNTHELABO (FR) 2000-08-09 EP disclosed
US-5719308-A Enzymatic process for the preparation of optically active tetralin derivatives SANOFI (FR) 1998-02-17 US disclosed
US-5573949-A Enzymatic process for the preparation of optically active Tetrahydro-2-naphthoic acids SANOFI (FR) 1996-11-12 US disclosed
EP-0683236-A1 Enzymatic process for the preparation of optical active tetralin-derivatives SANOFI (FR) 1995-11-22 EP disclosed