SCHEMBL8074469

SCHEMBL8074469

CC(C)(C#N)c1cc(CCl)cc(C(C)(C)C#N)c1F

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.36
UGT1A4 P22310 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3173073 0.80 CYP19A1 (0.49) CYP19A1UGT1A4PDE4D
SCHEMBL3866351 0.71 CA2 (0.34)
SCHEMBL12908860 0.69 CYP19A1 (0.40) CYP19A1UGT1A4PDE4D
SCHEMBL8583638 0.69
SCHEMBL13686005 0.68
SCHEMBL1041157 0.67 CYP19A1 (0.37) CYP19A1UGT1A4PDE4D
SCHEMBL12344152 0.66 CYP2A6 (0.37) CYP19A1UGT1A4PDE4D
SCHEMBL8069078 0.65 CYP19A1 (0.46) CYP19A1UGT1A4PDE4D
SCHEMBL26728887 0.65 ADORA1 (0.38)
SCHEMBL308410 0.65 NSD2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36617-E Anastrozole and salts as anticancer agent ZENECA LIMITED (GB) 2000-03-14 US disclosed
US-4935437-A (Substituted aralkyl) heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-19 US disclosed
EP-0296749-A1 (Substituted aralkyl) heterocyclic compounds ZENECA LIMITED (GB) 1988-12-28 EP disclosed