SCHEMBL8074993

SCHEMBL8074993

COc1ccc(CCN(CCO)CCO)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
BLM P54132 1/20 0.63
PMP22 Q01453 1/20 0.63
AOC3 Q16853 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.55
ATM Q13315 2/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54
KDM4E B2RXH2 1/20 0.54
SIGMAR1 Q99720 2/20 0.53
EBP Q15125 1/20 0.53
TMEM97 Q5BJF2 1/20 0.53
CA2 P00918 1/20 0.52
POLB P06746 1/20 0.51
CYP19A1 P11511 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088182 0.90 CYP1A2 (0.57) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL6574463 0.85 CYP3A4 (0.84) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL10959196 0.85 SIGMAR1 (0.70) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL21623605 0.83 CYP1A2 (0.69) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL29446268 0.82 ATM (0.66) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL13098004 0.82 ATM (0.66) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL13098012 0.82 ATM (0.66) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL296593 0.82 ATM (0.66) CYP1A2CYP3A4CYP2D6BLMPMP22
Hydrochloric Acid SCHEMBL8086550 0.82 BLM (0.66) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL9054003 0.82 SIGMAR1 (0.47) CYP1A2CYP3A4CYP2D6BLMPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711763-B1 1,4-DI(PHENYLALKYL)PIPERAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO LTD (JP) 2000-10-18 EP disclosed
US-5736546-A BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS SANTEN PHARMACEUTICAL CO., LTD. (JP) 1998-04-07 US disclosed
EP-0711763-A1 NOVEL 1,4-DI(PHENYLALKYL)PIPERAZINE DERIVATIVE SANTEN PHARMACEUTICAL CO., LTD. (JP) 1996-05-15 EP disclosed
EP-0388081-B1 Agent for the treatment of disorders of the cerebral neurotransmitter system SANTEN PHARMACEUTICAL CO LTD (JP) 1995-12-27 EP disclosed
US-5153198-A Fluoro-diphenylethylpiperazine for treating nervous system and brain disorders SANTEN PHARMACEUTICAL CO., LTD. (JP) 1992-10-06 US disclosed
US-5087627-A Administering diphenylethylpiperazine derivatives SANTEN PHARMACEUTICAL CO., LTD. (JP) 1992-02-11 US disclosed
EP-0388081-A2 Agent for the treatment of disorders of the cerebral neurotransmitter system SANTEN PHARMACEUTICAL CO., LTD. (JP) 1990-09-19 EP disclosed