SCHEMBL8075715

SCHEMBL8075715

CN(C)Cc1ccc(Cn2cc(C3=C(c4cn(C)c5ccccc45)C(=O)NC3=O)c3ccccc32)cc1

nearest known ligand 0.79

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 4/20 0.68
PIM1 P11309 2/20 0.68
PRKACA P17612 1/20 0.68
PRKACG P22612 1/20 0.68
PRKACB P22694 1/20 0.68
CDK2 P24941 3/20 0.65
PRKCB P05771 2/20 0.65
PRKCH P24723 2/20 0.65
PRKCE Q02156 2/20 0.65
PRKCQ Q04759 2/20 0.65
PRKCD Q05655 2/20 0.65
CCNE2 O96020 2/20 0.63
CDK4 P11802 2/20 0.63
CCND1 P24385 2/20 0.63
CCNE1 P24864 2/20 0.63
CAMK2D Q13557 1/20 0.61
GSK3B P49841 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065304 0.91 PRKCA (0.64) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8167903 0.89 CCNE2 (0.72) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8075459 0.87 PIM1 (0.70) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8073838 0.87 CCNE2 (0.66) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8122815 0.83 PRKCA (0.87) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL7057981 0.81 PRKCA (1.00) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8166825 0.81 SIRT2 (0.68) PIM1CDK2CCNE2CDK4CCND1
Hydrochloric Acid SCHEMBL8154146 0.80 PRKCA (0.98) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8072942 0.80 CCNE2 (0.62) PRKCAPIM1PRKACAPRKACGPRKACB
SCHEMBL8065185 0.80 PRKCA (0.68) PRKCAPIM1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153641-A Pharmaceutically active compounds ASTRA AKTIEBOLAG (SE) 2000-11-28 US disclosed