SCHEMBL807582

SCHEMBL807582

CCC[C@@H]1CCCN(Cc2cccc3cnccc23)C1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
MAPT P10636 1/20 0.56
HTT P42858 1/20 0.56
ROCK2 O75116 17/20 0.52
ROCK1 Q13464 7/20 0.52
TSHR P16473 1/20 0.48
CCR2 P41597 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084364 0.84 GAA (0.60) GAAMAPTHTTROCK2ROCK1
SCHEMBL15081998 0.81 GAA (0.57) GAAMAPTHTTROCK2ROCK1
SCHEMBL13754467 0.78 CACNA1B (0.66) GAAMAPTHTTROCK2ROCK1
SCHEMBL14193581 0.76 ROCK2 (0.57) GAAMAPTHTTROCK2ROCK1
SCHEMBL14193590 0.76 ROCK2 (0.57) GAAMAPTHTTROCK2ROCK1
SCHEMBL14193591 0.74 PRKD3 (0.56) GAAMAPTHTTROCK2ROCK1
SCHEMBL13595600 0.74 PRKD3 (0.56) GAAMAPTHTTROCK2ROCK1
SCHEMBL14193586 0.74 PRKD3 (0.56) GAAMAPTHTTROCK2ROCK1
SCHEMBL14193587 0.74 CXCR4 (0.53) GAAMAPTHTTROCK2ROCK1
SCHEMBL13595857 0.74 GAA (0.49) GAAMAPTHTTROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed