SCHEMBL8076292

SCHEMBL8076292

CCCC[C@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 16/20 0.48
CTSS P25774 1/20 0.46
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA7 P43166 1/20 0.41
CA14 Q9ULX7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8076295 1.00 CTSK (0.48) CTSKCTSSCA12CA1CA7
SCHEMBL4785511 0.95 CTSK (0.43) CTSKCTSS
SCHEMBL6333383 0.89 KDM4E (0.38) CTSKCTSSCA1CA7
SCHEMBL6333389 0.89 KDM4E (0.38) CTSKCTSSCA1CA7
SCHEMBL6333387 0.89 KDM4E (0.38) CTSKCTSSCA1CA7
SCHEMBL15344694 0.89 PLA2G2C (0.42) CTSKCTSS
SCHEMBL18648414 0.88 CTSK (0.47) CTSKCTSSCA12CA1CA7
SCHEMBL22722968 0.88 CTSK (0.47) CTSKCTSSCA12CA1CA7
SCHEMBL2013068 0.87 CA1 (0.44) CTSKCTSSCA12CA1CA7
SCHEMBL3178776 0.86 MEN1 (0.54) CTSKCTSSCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0555537-B1 Endothelin antagonists BANYU PHARMA CO LTD (JP) 2000-11-02 EP disclosed
US-5614498-A OLIGOPEPTIDES, BRONCHDILATORS BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-03-25 US disclosed
US-5496928-A Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
EP-0555537-A2 Endothelin antagonistic substance BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-18 EP disclosed