SCHEMBL807656

SCHEMBL807656

C/N=C(\C1=C(N)CCN(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2)C1)c1ccncc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 11/20 0.47
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HPGDS O60760 1/20 0.41
HDAC4 P56524 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PARP1 P09874 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
FPR3 P25089 1/20 0.38
FPR2 P25090 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL242088 0.76 USP30 (0.68) USP30HDAC4HDAC6PARP1GPR119
SCHEMBL242087 0.76 USP30 (0.68) USP30HDAC4HDAC6PARP1GPR119
SCHEMBL6200199 0.70 USP30 (0.69) USP30HDAC4HDAC6PARP1GPR119
SCHEMBL6200204 0.70 USP30 (0.69) USP30HDAC4HDAC6PARP1GPR119
SCHEMBL28975873 0.69 HDAC4 (0.60) USP30HDAC4HDAC6PARP1NPC1
SCHEMBL640458 0.69 ALDH1A1 (0.61) USP30NPC1RAB9AGPR119FPR3
SCHEMBL640457 0.69 ALDH1A1 (0.61) USP30NPC1RAB9AGPR119FPR3
SCHEMBL807196 0.68
SCHEMBL18741673 0.67 USP30 (0.51) USP30PARP1NPC1RAB9AGPR119
SCHEMBL18741675 0.67 USP30 (0.51) USP30PARP1NPC1RAB9AGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed