SCHEMBL8076891

SCHEMBL8076891

COC(=O)c1ncc(NC2CCNCC2)nc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.46
CDK1 P06493 1/20 0.46
CDK4 P11802 1/20 0.46
CCND1 P24385 1/20 0.46
HRH3 Q9Y5N1 2/20 0.45
HRH4 Q9H3N8 1/20 0.42
PDGFRB P09619 5/20 0.41
PDGFRA P16234 5/20 0.41
CLK2 P49760 2/20 0.41
CLK3 P49761 2/20 0.41
DYRK1A Q13627 2/20 0.41
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 1/20 0.39
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
CCNA2 P20248 1/20 0.38
IRAK4 Q9NWZ3 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR2C P28335 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2416166 0.76 PCSK9 (0.56) CDK2CDK1CDK4CCND1HRH3
SCHEMBL8061114 0.76 CDK2 (0.42) CDK2CDK1CDK4CCND1HRH3
Hydrochloric Acid SCHEMBL2416162 0.75 PCSK9 (0.55) CDK2CDK1CDK4CCND1HRH3
SCHEMBL14961898 0.75 PDGFRB (0.46) PDGFRBPDGFRAEGFRINSRLCK
SCHEMBL4233677 0.74 HCAR3 (0.56) CDK2CDK1CDK4CCND1HRH3
SCHEMBL614867 0.73 ATR (0.47) CDK2CDK1CDK4CCND1HRH4
SCHEMBL8077031 0.72 KDM4E (0.55)
SCHEMBL12248189 0.72 NPSR1 (0.47) IRAK4
SCHEMBL31584450 0.72 ATR (0.42)
SCHEMBL30062337 0.70 PRMT5 (0.48) HRH3HRH4CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156758-A Antibacterial quinazoline compounds ISIS PHARMACEUTICALS, INC. (US) 2000-12-05 US disclosed