SCHEMBL8077008

SCHEMBL8077008

CC1=C(n2cc(Br)cc(N)c2=O)c2cc([N+](=O)[O-])ccc2OC1(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.39
CYP3A4 P08684 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.35
MEN1 O00255 5/20 0.35
KMT2A Q03164 5/20 0.35
POLB P06746 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
CASP1 P29466 1/20 0.32
CASP3 P42574 1/20 0.32
CASP4 P49662 1/20 0.32
CASP7 P55210 1/20 0.32
CASP9 P55211 1/20 0.32
CASP6 P55212 1/20 0.32
HTT P42858 1/20 0.32
PTPRC P08575 1/20 0.32
S100A4 P26447 1/20 0.32
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
CHRM2 P08172 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8189795 0.90 MEN1 (0.36) TDP1CYP3A4ALDH1A1TSHRMEN1
SCHEMBL8084356 0.89 MEN1 (0.35) TDP1CYP3A4ALDH1A1MEN1KMT2A
SCHEMBL8088643 0.88 CYP3A4 (0.36) TDP1CYP3A4ALDH1A1TSHRMEN1
SCHEMBL8088765 0.86 CYP3A4 (0.36) TDP1CYP3A4ALDH1A1TSHRMEN1
SCHEMBL8085265 0.84 MEN1 (0.35) TDP1CYP3A4ALDH1A1TSHRMEN1
SCHEMBL8076907 0.83 TDP1 (0.37) TDP1CYP3A4ALDH1A1TSHRMEN1
SCHEMBL8085097 0.83 CFTR (0.38) ALDH1A1MEN1KMT2AHTT
SCHEMBL8088721 0.82 MALT1 (0.33) MALT1CASP3
SCHEMBL8077044 0.82 PDE7A (0.34) TDP1CYP3A4ALDH1A1TSHRMEN1
SCHEMBL8076960 0.81 MEN1 (0.37) TDP1CYP3A4ALDH1A1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed