SCHEMBL8078336

SCHEMBL8078336

C=C(CCCCCNC(=O)C(=O)c1cn2c3c(cccc13)CCC2)NOCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.43
MTNR1B P49286 7/20 0.43
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
PREP P48147 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3057715 0.92 MTNR1A (0.47) MTNR1AMTNR1BHTR2AHTR2C
SCHEMBL3053168 0.91 MTNR1A (0.47) MTNR1AMTNR1BHTR2AHTR2CALDH1A1
SCHEMBL3058587 0.88 MTNR1A (0.48) MTNR1AMTNR1BHTR2AHTR2CALDH1A1
SCHEMBL3053598 0.83 MTNR1A (0.53) MTNR1AMTNR1BHTR2AHTR2CALDH1A1
SCHEMBL3060093 0.83 MTNR1A (0.48) MTNR1AMTNR1BALDH1A1KDM4EMEN1
SCHEMBL3058774 0.82 MTNR1A (0.49) MTNR1AMTNR1BALDH1A1HTTKDM4E
SCHEMBL3053869 0.81 MTNR1A (0.52) MTNR1AMTNR1BHTR2AHTR2CALDH1A1
SCHEMBL3056854 0.80 MTNR1A (0.53) MTNR1AMTNR1BALDH1A1KDM4EMEN1
SCHEMBL3054181 0.80 MTNR1A (0.53) MTNR1AMTNR1BALDH1A1KDM4EMEN1
SCHEMBL3052990 0.80 MTNR1A (0.48) MTNR1AMTNR1BALDH1A1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026446-A9 HDAC INHIBITORS ARQULE, INC. (US) 2010-03-11 WO disclosed
WO-2009026446-A2 HDAC INHIBITORS ARQULE, INC. (US) 2009-02-26 WO disclosed